Compound | Mode of inhibition | Ki (μM) | Km (μM) |
---|---|---|---|
18 | Uncompetitive | 21.08 ± 12.25 | 0.12 ± 0.03 |
5 | Noncompetitive | 39.88 ± 8.47 | 0.14 ± 0.01 |
8 | Competitive | 11.16 ± 0.99 | 0.18 ± 0.01 |
6 | Mixed | 57.76 ± 1.67 | 0.17 ± 0.01 |
9 | Mixed | 54.42 ± 15.76 | 0.17 ± 0.01 |
22 | Mixed | 7.00 ± 1.97 | 0.04 ± 0.01 |
24 | Mixed | 43.96 ± 0.88 | 0.08 ± 0.01 |