Crude extract | Babesia and Theileria | IC50 (μg/mL)a | EC50 (μg/mL)b | Selective indices c | ||||
---|---|---|---|---|---|---|---|---|
MDBK | NIH/3 T3 | HFF | MDBK | NIH/3 T3 | HFF | |||
MEVT | B. bovis | 75.7 ± 2.6 | 930 ± 29.9 | 1260 ± 18.9 | >1500 | 12.3 | 16.7 | > 19.8 |
B. bigemina | 43.3 ± 1.8 | 930 ± 29.9 | 1260 ± 18.9 | >1500 | 21.5 | 29.1 | > 34.6 | |
B. divergens | 67.6 ± 2.8 | 930 ± 29.9 | 1260 ± 18.9 | >1500 | 13.8 | 18.6 | > 22.2 | |
B. caballi | 48 ± 3.8 | 930 ± 29.9 | 1260 ± 18.9 | >1500 | 19.4 | 26.3 | > 31.3 | |
T. equi | 54 ± 2.1 | 930 ± 29.9 | 1260 ± 18.9 | >1500 | 17.2 | 23.3 | > 27.8 | |
AELN | B. bovis | 86.6 ± 8.2 | 573.7 ± 12.4 | 831 ± 19.9 | >1500 | 6.6 | 9.6 | > 17.3 |
B. bigemina | 33.3 ± 5.1 | 573.7 ± 12.4 | 831 ± 19.9 | >1500 | 17.2 | 25 | > 45.1 | |
B. divergens | 62.2 ± 3.3 | 573.7 ± 12.4 | 831 ± 19.9 | >1500 | 9.2 | 13.4 | > 24.1 | |
B. caballi | 34.5 ± 7.5 | 573.7 ± 12.4 | 831 ± 19.9 | >1500 | 16.6 | 24.1 | > 43.5 | |
T. equi | 82.2 ± 9.3 | 573.7 ± 12.4 | 831 ± 19.9 | >1500 | 7 | 10.1 | > 18.2 |