Skeleton | Compounds | Binding site in CDK2 | Binding site in CDK6 |
---|---|---|---|
Lupane-type | LF01 | hinge residues, catalytic loop | catalytic loop |
LF04 | hinge residues | catalytic loop, activation segment | |
LF08 | Â | catalytic loop, activation segment | |
LF09 | K of K/E/D/D | catalytic loop | |
LFa | hinge residues, K of K/E/D/D | catalytic loop | |
Oleanane-type | LF02 | K of K/E/D/D | catalytic loop |
LF03 | hinge residues, K of K/E/D/D | catalytic loop | |
LF05 | hinge residues, catalytic loop, activation segment | catalytic loop | |
LF07 | hinge residues | catalytic loop | |
LF10 | hinge residues | catalytic loop, activation segment | |
LF11 | hinge residues | catalytic loop, activation segment | |
LF12 | hinge residues, K of K/E/D/D | catalytic loop | |
LF13 | hinge residues, K of K/E/D/D | catalytic loop | |
LFb | hinge residues, K of K/E/D/D, catalytic loop | catalytic loop | |
LFc | hinge residues, K of K/E/D/D, catalytic loop | Â | |
LFd | Â | catalytic loop | |
LFe | catalytic loop, activation segment | activation segment | |
LFf | K of K/E/D/D, catalytic loop | activation segment | |
Ursane-type | LF06 | Â | activation segment |
LFg | hinge residues, K of K/E/D/D | catalytic loop |