Extracts | Brine shrimp cytotoxicity | THP-1 cytotoxicity | Hep G2 cytotoxicity | Protein kinase inhibition | |||||
---|---|---|---|---|---|---|---|---|---|
% mortality | LC50 (μg/ml) | % inhibition | IC50(μg/ml) | % inhibition | IC50 (μg/ml) | Diameter (mm) at 100 μg/disc | MIC (μg/disc) | ||
200 μg/ml | 20 μg/ml | 20 μg/ml | Clear zone | Bald zone | |||||
Nh | 63.33 ± 5.77bc | 91.40 ± 0.23 | 31.5 ± 1.5 | > 20 | 61.14 ± 0.70c | 8.95 ± 0.20 | 10.00 ± 1.0 | 16.00 ± 1.0e | 12.5 |
Nh-Ea | 73.33 ± 5.77b | 112.37 ± 1.20 | 45.57 ± 1.00c | > 20 | 38.43 ± 0.78 | > 20 | 6.67 ± 0.58 | 9.67 ± 0.58 | 100 |
Nh-E | 53.33 ± 5.77cd | 153.33 ± 1.12 | 35.87 ± 0.85 | > 20 | 57.37 ± 0.67d | 19.10 ± 0.50 | 6.67 ± 0.58 | 15.00 ± 1.0e | 25 |
C | 93.33 ± 5.77a | 85.40 ± 0.26 | 26.67 ± 0.91 | > 20 | 60.50 ± 0.50c | 9.50 ± 0.28 | 6.67 ± 0.58 | 10.67 ± 0.58fg | 50 |
Ea | 43.33 ± 5.77 | > 200 | 14.17 ± 1.35 | > 20 | 61.53 ± 0.35c | 8.63 ± 0.30 | 6.67 ± 0.58 | 9.33 ± 0.58 | 100 |
C-M | 53.33 ± 5.77cd | > 200 | 18.27 ± 2.91 | > 20 | 20.60 ± 0.30 | > 20 | 9.00 ± 1.0 | 12.00 ± 1.0f | 100 |
Ea-M | 63.33 ± 5.77bc | 137.37 ± 0.55 | 19.63 ± 2.87 | > 20 | 31.45 ± 0.15 | > 20 | 9.00 ± 1.0 | 30.00 ± 1.0b | 12.5 |
A | 63.33 ± 5.77bc | 123.83 ± 0.95 | 33.13 ± 1.70 | > 20 | 54.71 ± 0.25e | 19.80 ± 0.20 | – | 12.00 ± 1.0f | 100 |
M | 93.33 ± 5.77a | 110 ± 0.75 | 45.37 ± 1.56c | > 20 | 56.63 ± 0.20d | 19.76 ± 0.20 | 28 ± 1.0 | 40.00 ± 1.0a | 12.5 |
A-M | 63.33 ± 5.77bc | 123.5 ± 0.92 | 77.63 ± 1.33b | 4.9 ± 0.20 | 25.90 ± 0.19 | > 20 | 15.00 ± 1.0 | 25.0 ± 1.0c | 50 |
A-E | 93.33 ± 5.77a | 123.4 ± 0.89 | 48.27 ± 3.00c | > 20 | 49.80 ± 0.67 | > 20 | 6.67 ± 0.58 | 12.0 ± 1.0f | 100 |
E | 96.67 ± 5.77a | 46.91 ± 0.19 | 20.8 ± 1.90 | > 20 | 37.40 ± 0.30 | > 20 | 6.33 ± 0.58 | 7.67 ± 0.58 | – |
A-Dw | 93.33 ± 5.77a | 52.63 ± 1.11 | 47.43 ± 2.16c | > 20 | 29.60 ± 0.80 | > 20 | 7.00 ± 1.0 | 15.00 ± 1.0e | 50 |
M-Dw | 93.33 ± 5.77a | 64.93 ± 1.40 | 30.47 ± 1.95 | > 20 | 63.07 ± 0.40b | 8.68 ± 0.25 | – | 12.00 ± 1.0f | 100 |
Dw | 33.33 ± 5.77 | > 200 | 36.7 ± 1.15 | > 20 | 46.83 ± 0.25 | > 20 | 7.00 ± 1.0 | – | – |
Doxorubicin | 96.67 ± 5.77a | 5.63 ± 0.25 |  |  | 98.37 ± 0.15a | 5.30 ± 0.20 |  |  |  |
5-Florouracil |  |  | 99.2 ± 0.92a | 5.13 ± 0.13 |  |  |  |  |  |
Vincristine |  |  | 99.33 ± 0.83a | 8.24 ± 0.12 |  |  |  |  |  |
Surfactin |  |  |  |  |  |  |  | 20 ± 1.0d |  |
DMSO | – |  | – |  | – |  |  | – |  |