Samples | Cytotoxicty (LC50, μg/ml) | Selectivity indexa | |||||||
---|---|---|---|---|---|---|---|---|---|
 | C.a | C.A | A.f | C.n | S.a | P.a | E.f | E.c | |
Extract and fractions | Â | Â | Â | Â | Â | Â | Â | Â | Â |
Crude extract | 53.45 ± 2.21 | 0.04 | 0.04 | 0.21* | 0.08 | 0.67 | 0.17 | 0.67 | 0.67 |
Fraction A | 17.91 ± 1.71 | 0.03 | 0.09* | 0.05* | 0.01 | 0.90 | 0.06 | 0.45 | 0.45 |
Fraction B | 93.76 ± 25.62 | 0.08 | 0.22* | 0.66* | 0.66* | 0.59 | 0.30 | 1.17 | 1.17 |
Compounds | Â | Â | Â | Â | Â | Â | Â | Â | Â |
Robusflavone A (1) | 13.20 ± 0.02 | 0.05 | 0.20 | 0.16* | 0.05 | 0.05 | 0.21 | 0.05 | 0.05 |
Robusflavone B (2) | 30.42 ± 3.26 | 0.24 | 0.47 | 0.36* | 0.47 | 0.24 | 0.48 | 0.48 | 0.24 |
Orostachyscerebroside A (3) | > 100 | 0.4 | 0.53* | 0.53* | 0.4 | 0.8 | 1.59 | 0.8 | 0.8 |
Stigmasterol (4) | 54.97 ± 11.05 | 0.44 | 0.44 | 0.85 | 0.44 | 0.44 | 0.87 | 0.22 | 0.22 |
1-O-Heptatriacontanoylglycerol (5) | 91.52 ± 28.38 | 0.37 | 1.41 | 0.73 | 0.37 | 0.73 | 1.45 | 0.73 | 0.73 |
Eicosanoic acid (6) | NT | - | - | - | - | - | - | - | - |
3-O-β-D-Glucopyranoside of sitosterol (7) | >100 | 0.80 | 0.80 | 1.17* | 1.17* | 0.80 | 1.58 | 1.58 | 0.80 |
6-Prenylpinocembrin (8) | 21.87 ± 0.37 | 0.17 | 0.34 | 0.13* | 0.09 | 0.70 | 0.35 | 0.35 | 0.35 |
Control | Â | Â | Â | Â | Â | Â | Â | Â | Â |
Dox | 3.32 ± 1.31 |  |  |  |  |  |  |  |  |